GSK6853
Supplier:
Catalogue number:
10-4016-01
Size:
5 mg
Product is available in:
BRPF1 inhibitor / Very potent (pIC50 = 8.6 vs full length protein, 7.7 in cellular assays) inhibitor of Bromodomain and PHD Finger-containing 1 (BRPF1). It displayed >1600-fold selectivity over other bromodomains.
Product Type:
Biochemicals & reagents
CAS Number:
1910124-24-1
Reference:
Bamborough et al. (2016), GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain; ACS Med.Chem. Lett. 7 552
Storage Temperature:
-20°C
Additional Information:
TARGET: Bromodomain -- PATHWAY: Chromatin -- RESEARCH AREA: Epigenetics